Antitrypanosomal activity of 5-nitro-2-aminothiazole-based compounds
نویسندگان
چکیده
منابع مشابه
Antitrypanosomal activity of 5-nitro-2-aminothiazole-based compounds
A small series of 5-nitro-2-aminothiazole-based amides containing arylpiperazine-, biphenyl- or aryloxyphenyl groups in their core were synthesized and evaluated as antitrypanosomatid agents. All tested compounds were active or moderately active against Trypanosoma cruzi amastigotes in infected L6 cells and Trypanosoma brucei brucei, four of eleven compounds were moderately active against Leish...
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ژورنال
عنوان ژورنال: European Journal of Medicinal Chemistry
سال: 2016
ISSN: 0223-5234
DOI: 10.1016/j.ejmech.2016.04.010